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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T12829 | Salmeterol | GR33343X | Adrenergic Receptor |
Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma. | |||
T3284 | Carazolol | Conducton,Suacron | Adrenergic Receptor |
Carazolol (Suacron) is a high-affinity antagonist/partial inverse agonist (also referred to as a beta blocker) of the β-adrenergic receptor. | |||
T1584 | Terbutaline Sulfate | Terbutaline hemisulfate | Antibacterial , Adrenergic Receptor , Antibiotic |
Terbutaline Sulfate (Terbutaline hemisulfate) is a selective beta-2 adrenergic agonist used as a bronchodilator and tocolytic. | |||
T4983 | Isoetharine mesylate salt | Isoetarine mesilate | Others , Adrenergic Receptor |
Isoetharine mesylate salt (Isoetarine mesilate) is a β-adrenergic receptor agonist. it also is pregnane X receptor (PXR) activator capable of upregulating CYP450 expression. | |||
T6653 | Salmeterol Xinafoate | Salmetedur,GR 33343X xinafoate,Arial | HIV Protease , Adrenergic Receptor |
Salmeterol Xinafoate (GR 33343X xinafoate) is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma symptoms and chronic obstructive pulmonary disease (COPD) symptom... | |||
T13403 | ZK-90055 hydrochloride | ZK 90055 hydrochloride,ZK90055 hydrochloride | Adrenergic Receptor |
ZK-90055 hydrochloride is a β2 adrenergic receptor agonist used to study asthma. | |||
T40622 | Mapenterol hydrochloride | Adrenergic Receptor | |
Mapenterol hydrochloride is an agonist of β2-adrenergic receptor. | |||
T6522 | Guanabenz Acetate | Wy8678 acetate,BR-750,Wytensin | Adrenergic Receptor |
Guanabenz Acetate (Wytensin) is a specific agonist of adrenergic receptor. The pEC50 for α2a-adrenergic receptor, α2b-adrenergic receptor and α2c-adrenergic receptor is 8.25, 7.01 and ~5, respectively. | |||
T4548 | Procaterol hydrochloride | Adrenergic Receptor | |
Short-acting β2-adrenergic receptor agonist used to treat asthma. | |||
T15819 | LY377604 | Adrenergic Receptor | |
LY377604 is a human β3-adrenergic receptor agonist (EC50: 2.4 nM) and β1/2-adrenergic receptor antagonist for the study of obesity. | |||
T7065 | Tizanidine | Adrenergic Receptor | |
Tizanidine, an α2-adrenergic receptor agonist, suppresses the release of neurotransmitters from central nervous system (CNS) noradrenergic neurons. | |||
T26119 | Romifidine | Romifidinum | |
Romifidine is used as a sedative in veterinary medicine mainly in large animals such as horses. It acts as an agonist at the α2 adrenergic receptor subtype. | |||
T10052 | AR-08 | Adrenergic Receptor | |
T68023L | Tolnapersine TFA | Tolnapersine TFA(70312-00-4 Free base) | Dopamine Receptor , Adrenergic Receptor |
Tolnapersine TFA is a mixed dopamine agonist and alpha adrenergic receptor antagonist. | |||
T34256 | Rafabegron | TAK-677,TAK677,AD9677,AD-9677,TAK 677,AD 9677 | Adrenergic Receptor |
Rafabegron (TAK677) is a potent and selective β3 adrenergic receptor agonist for the study of diabetes and obesity. | |||
T6652 | Salbutamol hemisulfate | Ventolin Sulfate,Albuterol,Salbutamol Sulfate,Bronchospray,Albuterol Sulfate | Adrenergic Receptor , Autophagy |
Salbutamol hemisulfate (Albuterol Sulfate) is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 μM. | |||
T33386 | Milveterol HCl | Milveterol,GSK-159797,GSK 159797,GSK159797 | Adrenergic Receptor |
Milveterol HCl is a long-acting β(2) -adrenergic receptor agonist for the potential treatment of chronic obstructive pulmonary disease (COPD). | |||
T21371 | Apraclonidine hydrochloride | Iopidine,ALO 2145,Apraclonidina,P-aminoclonidine,4-Aminoclonidine,Apraclonidine HCl,Apraclonidinum | Adrenergic Receptor |
Apraclonidine hydrochloride (ALO 2145) is an α2-adrenergic agonist and a weak α-1 adrenergic receptor agonist. Apraclonidine hydrochloride lowers intraocular pressure in human eyes and can be used in studies about glauco... | |||
T6422 | Brimonidine Tartrate | AGN190342 tartrate,304 tartrate,AGN190342 (tartrate),UK 14304 (tartrate),UK14304 tartrate | Adrenergic Receptor |
Brimonidine Tartrate (AGN190342 tartrate) is a quinoxaline derivative and adrenergic α-2 receptor agonist (EC50: 0.45 nM) that is used to manage intraocular pressure associated with open-angle glaucoma or ocular hyperten... | |||
T68114L | Nardeterol HCl | Nardeterol HCl(73865-18-6 Free base) | Adrenergic Receptor |
Nardeterol HCl is a β-adrenergic receptor partial agonist used in the study of the central nervous system.CAS 번호13460-73-83-4 | |||
T23397 | ST 91 | Others , Adrenergic Receptor | |
ST-91 is an agonist of α2-adrenoceptor with a mixed α-adrenergic receptor type/subtype selection profile. | |||
T31750 | Faxeladol | EM906,GCR 9905,EM 906,GCR-9905,EM-906,GCR9905 | 5-HT Receptor , Opioid Receptor , Adrenergic Receptor |
Faxeladol, a potent adrenergic absorption inhibitor and serotonin reuptake inhibitor, is a small-molecule Opioid receptor agonist that can be used to study neurological disorders. | |||
T8810 | Terbutaline | Adrenergic Receptor | |
Terbutaline is a short-acting agonist of β2-adrenergic receptor (β2-AR) . It is an active metabolite of bambuterol | |||
T7164 | Levalbuterol tartrate | Levosalbutamol tartrate | Adrenergic Receptor |
Levalbuterol tartrate (Levosalbutamol tartrate) is the β2-adrenergic receptor agonist,and is used to treatment of asthma. | |||
T8358 | Fenoterol | Adrenergic Receptor | |
Fenoterol is an agonist of β2-adrenergic receptor It is classed as sympathomimetic beta agonist and asthma medication. | |||
T5954 | Methyldopa hydrate | Alpha-Methyldopa Sesquihydrate,L-(-)-α-Methyldopa hydrate,MK-351 hydrate,Methyldopa Sesquihydrate | Dopamine Receptor , Adrenergic Receptor |
Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension. It inhibits the sympathetic nervous system, decreases production of dopamine, ... | |||
T22612 | BMY-14802 hydrochloride | BMS 181100 hydrochloride,BMY-14802-1,BMY 14802 hydrochloride | Sigma receptor , 5-HT Receptor , Adrenergic Receptor |
BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 nM) with antipsychotic effects. BMY-14802 hydrochloride is an agonist of the α1-adrenergic receptor and 5-HT1A. | |||
T0290 | Tizanidine hydrochloride | Tizanidine HCl,DS 103-282 | Adrenergic Receptor |
Tizanidine hydrochloride (Tizanidine HCl), an α2-adrenergic receptor agonist, inhibits neurotransmitter release from CNS noradrenergic neurons. | |||
T11318 | Dopexamine hydrochloride | FPL60278AR | Adrenergic Receptor |
Dopexamine hydrochloride (FPL60278AR) is a β2-adrenergic receptor agonist. Dopexamine can attenuate the inflammatory response and protect against organ injury in the absence of significant effects on hemodynamics or regi... | |||
T22871 | Ipsapirone | 5-HT Receptor | |
Ipsapirone is a partial agonist of 5-HT1A receptor and produces an inhibitory effect on 5-HT2 and the α1-adrenergic function at high doses. | |||
T10952 | Dabuzalgron | Ro 115-1240 | Apoptosis , Adrenergic Receptor |
Dabuzalgron (Ro 115-1240) is an orally active selective alpha-1A adrenergic receptor agonist used to treat urinary incontinence. Dabuzaron prevents cardiotoxicity caused by doxorubicin by maintaining mitochondrial functi... | |||
T3277 | Tulobuterol hydrochloride | Lobuterol,Hokunalin,Berachin | Influenza Virus , Adrenergic Receptor , Antibiotic |
Tulobuterol hydrochloride (Hokunalin) is a long-acting beta2-adrenergic receptor agonist. | |||
T3046 | BMY 7378 dihydrochloride | BMY7378 HCl | Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor |
BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor. | |||
T21447 | Tolazoline | Priscol,Priscoline,Pridazole,Divascol,Vasimid,Benzalolin | Adrenergic Receptor |
Tolazoline (Benzalolin), a non-selective competitive α-adrenergic receptor antagonist, is used as a vasodilator to treat spasms of peripheral blood vessels. It has also been used successfully as an antidote to reverse th... | |||
T6703 | Tetrahydrozoline hydrochloride | Murine Plus,Tetryzoline hydrochloride,Tyzine,Tetrahydrozoline HCl | Adrenergic Receptor |
Tetrahydrozoline hydrochloride (Murine Plus) is an imidazoline derivative with alpha receptor agonist activity. | |||
T22029 | AL 34662 | 5-HT Receptor , Adrenergic Receptor | |
AL 34662 is a selective and potent 5-HT2A receptor agonist with IC50s of 0.77 nM and 1.5 nM for rat and human 5-HT2 receptors, respectively.AL 34662 is also a low affinity α-1D adrenergic agonist, with an EC50 of 0.4 μM.... | |||
T2631 | WAY-100635 Monomaleate | Dopamine Receptor , 5-HT Receptor | |
WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM. It is also a dopamine D4 receptor agonist with pIC50 values of 8.9 and 6.6 for 5-HT1A ... | |||
T1735 | Lurasidone hydrochloride | Lurasidone HCl,SM-13496 (Hydrochloride),SM-13496 | Dopamine Receptor , 5-HT Receptor , Norepinephrine |
Lurasidone hydrochloride (Lurasidone HCl) is a thiazole derivative and atypical antipsychotic agent that functions as a dopamine D2 receptor antagonist; serotonin 5-HT2 receptor antagonist, serotonin 5-HT7 receptor antag... | |||
T12970 | Solabegron | GW 427353 | Adrenergic Receptor |
Solabegron (GW 427353) is a selective agonist of β3-adrenergic receptor, stimulating cAMP accumulation in Chinese hamster ovary cells expressing the human β3-AR(EC50 : 22 nM). It is used for treatment of overactive bladd... | |||
T6466 | Dexmedetomidine hydrochloride | Precedex,(+)-Medetomidine hydrochloride,(S)-Medetomidine hydrochloride,Dexmedetomidine HCl | Adrenergic Receptor |
Dexmedetomidine hydrochloride (Precedex) is an imidazole derivative that is an agonist of the adrenergic alpha-2 receptor. It is closely-related to MEDETOMIDINE, which is the racemic form of this compound. | |||
T23557 | Talibegron hydrochloride | ZD2079 hydrochloride,ZD 2079 | Adrenergic Receptor |
Talibegron hydrochloride (ZD2079 hydrochloride) is an β3 adrenergic receptor agonist with a pD2 of 3.72 on phenylephrine-preconstricted rat mesenteric artery. Relaxes rat mesenteric artery and isolated aorta in vitro. In... | |||
T26666 | ASM-024 | AChR | |
ASM-024, a potent nicotinic receptor agonist, is a small molecule synthetic piperazine compound that promotes different targets and signaling pathways of β2-adrenergic receptors mediating smooth muscle relaxation, and is... | |||
T68129L1 | Picumeterol FA | Picumeterol FA(130641-36-0 Free base) | Adrenergic Receptor |
picumeterol FA is a potent and selective β2-adrenergic receptor agonist. In in vitro and in vivo tests, picumeterol FA produces long-lasting airway smooth muscle relaxation. picumeterol FA is a pure R-enantiomer and can ... | |||
T38192 | Unifiram | Others | |
Unifiram is a nootropic agent.1It increases acetylcholine (ACh) release in the rat cerebral cortexin vivoand induces a long-lasting increase in the amplitude of field excitatory postsynaptic potentials (fEPSPs) in the ra... | |||
T24670 | Protokylol | JB-251,Protokylolum,JB 251,JB251,Protoquilol | |
Protokylol is a β-adrenergic receptor agonist. | |||
T25003 | Acrinor | H 835 | |
Acrinor is a adrenergic beta receptor agonist. | |||
T28885 | Sunepitron HCl | CP 93,393,CP93,393,CP-93393,CP93393,CP 93393,CP-93,393 | |
Sunepitron is a combined α2-adrenergic receptor antagonist and 5-HT1A receptor agonist. | |||
T11512 | Guanoxabenz | Hydroxyguanabenz | Others |
T23281 | RWJ 52353 | Others | |
α2D adrenergic receptor agonist | |||
T26651 | ARC-239 | ARC239,AR C 239,AR C239,AR C-239 | |
ARC-239 is an agonist of α2-adrenergic receptor. |
カタログ番号 | 製品名 | 別名 | ターゲット |
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T6688 | Synephrine hydrochloride | Oxedrine hydrochloride,Synephrine HCl | Endogenous Metabolite , Adrenergic Receptor |
Synephrine hydrochloride (Oxedrine hydrochloride) is an agonist that acts on sympathomimetic α-adrenergic receptor (AR). | |||
T0453 | Phenylephrine hydrochloride | NCI-c55641,Phenylephrine HCl,(R)-(-)-Phenylephrine hydrochloride | Endogenous Metabolite , Adrenergic Receptor |
Phenylephrine hydrochloride (NCI-c55641) is a selective agonist of the α1-adrenergic receptor. | |||
T4429 | Rauwolscine hydrochloride | Corynanthidine hydrochloride,α-Yohimbine hydrochloride,Isoyohimbine hydrochloride | Adrenergic Receptor |
Rauwolscine hydrochloride (Isoyohimbine hydrochloride) , a natural alkaloid, is a specific and reversible α2-adrenergic receptor antagonist (Ki: 12 nM) [1]. It is a stereoisomer of yohimbine, which potently antagonizes b... | |||
T6662 | Scopine | 6,7-Epoxytropine | Adrenergic Receptor |
Scopine (6,7-Epoxytropine), the metabolite of anisodine, is an α1-adrenergic receptor agonist used in the therapy of acute circulatory shock. | |||
TN1465 | Cannabigerol | NOS , 5-HT Receptor , ROS | |
Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; also binds to the CB2 receptor; it can relieve interocular pressur... | |||
T6519 | Gramine | NSC 16892,Donaxine | Adiponectin receptor , Reverse Transcriptase , Adrenergic Receptor |
Gramine (Donaxine), a natural indole alkaloid, present in several plant species, acts as an active adiponectin receptor (AdipoR) agonist, with IC50s of 3.2 and 4.2 μM for AdipoR2 and AdipoR1, respectively. Gramine is als... | |||
T8149 | Dobutamine hydrochloride | Dobutamine (hydrochloride) | Adrenergic Receptor |
Dobutamine hydrochloride (Dobutamine (hydrochloride)) is a catecholamine that acts as a β-adrenergic receptor agonist with potent positive inotropic effects. | |||
T60245 | Norepinephrine hydrochloride | ||
Norepinephrine hydrochloride (Levarterenol hydrochloride) is a β1 -selective agonist of the adrenergic receptor with EC 50 of 5.37 μM [1]. |
カタログ番号 | 製品名 | Species | Expression System |
---|---|---|---|
TMPJ-00983 | ARRB1 Protein, Human, Recombinant (His) | Human | E. coli |
β-Arrestin-1 (ARRB1) is a cytoplasmic protein that belongs to the arrestin family. ARRB1 is expressed at high levels in peripheral blood leukocytes and the central nervous system. ARRB1 regulates agonist-mediated G-prote... | |||
TMPH-02540 | GRK2 Protein, Mouse, Recombinant (His & SUMO) | Mouse | E. coli |
Specifically phosphorylates the agonist-occupied form of the beta-adrenergic and closely related receptors, probably inducing a desensitization of them. Key regulator of LPAR1 signaling. Competes with RALA for binding to... |