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Search Results for " adrenergic receptor agonist "

ターゲット

119

阻害剤

8

天然化合物

2

リコンビナントタンパク質

カタログ番号 製品名 別名 ターゲット
T12829 Salmeterol GR33343X Adrenergic Receptor
Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.
T3284 Carazolol Conducton,Suacron Adrenergic Receptor
Carazolol (Suacron) is a high-affinity antagonist/partial inverse agonist (also referred to as a beta blocker) of the β-adrenergic receptor.
T1584 Terbutaline Sulfate Terbutaline hemisulfate Antibacterial , Adrenergic Receptor , Antibiotic
Terbutaline Sulfate (Terbutaline hemisulfate) is a selective beta-2 adrenergic agonist used as a bronchodilator and tocolytic.
T4983 Isoetharine mesylate salt Isoetarine mesilate Others , Adrenergic Receptor
Isoetharine mesylate salt (Isoetarine mesilate) is a β-adrenergic receptor agonist. it also is pregnane X receptor (PXR) activator capable of upregulating CYP450 expression.
T6653 Salmeterol Xinafoate Salmetedur,GR 33343X xinafoate,Arial HIV Protease , Adrenergic Receptor
Salmeterol Xinafoate (GR 33343X xinafoate) is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma symptoms and chronic obstructive pulmonary disease (COPD) symptom...
T13403 ZK-90055 hydrochloride ZK 90055 hydrochloride,ZK90055 hydrochloride Adrenergic Receptor
ZK-90055 hydrochloride is a β2 adrenergic receptor agonist used to study asthma.
T40622 Mapenterol hydrochloride Adrenergic Receptor
Mapenterol hydrochloride is an agonist of β2-adrenergic receptor.
T6522 Guanabenz Acetate Wy8678 acetate,BR-750,Wytensin Adrenergic Receptor
Guanabenz Acetate (Wytensin) is a specific agonist of adrenergic receptor. The pEC50 for α2a-adrenergic receptor, α2b-adrenergic receptor and α2c-adrenergic receptor is 8.25, 7.01 and ~5, respectively.
T4548 Procaterol hydrochloride Adrenergic Receptor
Short-acting β2-adrenergic receptor agonist used to treat asthma.
T15819 LY377604 Adrenergic Receptor
LY377604 is a human β3-adrenergic receptor agonist (EC50: 2.4 nM) and β1/2-adrenergic receptor antagonist for the study of obesity.
T7065 Tizanidine Adrenergic Receptor
Tizanidine, an α2-adrenergic receptor agonist, suppresses the release of neurotransmitters from central nervous system (CNS) noradrenergic neurons.
T26119 Romifidine Romifidinum
Romifidine is used as a sedative in veterinary medicine mainly in large animals such as horses. It acts as an agonist at the α2 adrenergic receptor subtype.
T10052 AR-08 Adrenergic Receptor
T68023L Tolnapersine TFA Tolnapersine TFA(70312-00-4 Free base) Dopamine Receptor , Adrenergic Receptor
Tolnapersine TFA is a mixed dopamine agonist and alpha adrenergic receptor antagonist.
T34256 Rafabegron TAK-677,TAK677,AD9677,AD-9677,TAK 677,AD 9677 Adrenergic Receptor
Rafabegron (TAK677) is a potent and selective β3 adrenergic receptor agonist for the study of diabetes and obesity.
T6652 Salbutamol hemisulfate Ventolin Sulfate,Albuterol,Salbutamol Sulfate,Bronchospray,Albuterol Sulfate Adrenergic Receptor , Autophagy
Salbutamol hemisulfate (Albuterol Sulfate) is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 μM.
T33386 Milveterol HCl Milveterol,GSK-159797,GSK 159797,GSK159797 Adrenergic Receptor
Milveterol HCl is a long-acting β(2) -adrenergic receptor agonist for the potential treatment of chronic obstructive pulmonary disease (COPD).
T21371 Apraclonidine hydrochloride Iopidine,ALO 2145,Apraclonidina,P-aminoclonidine,4-Aminoclonidine,Apraclonidine HCl,Apraclonidinum Adrenergic Receptor
Apraclonidine hydrochloride (ALO 2145) is an α2-adrenergic agonist and a weak α-1 adrenergic receptor agonist. Apraclonidine hydrochloride lowers intraocular pressure in human eyes and can be used in studies about glauco...
T6422 Brimonidine Tartrate AGN190342 tartrate,304 tartrate,AGN190342 (tartrate),UK 14304 (tartrate),UK14304 tartrate Adrenergic Receptor
Brimonidine Tartrate (AGN190342 tartrate) is a quinoxaline derivative and adrenergic α-2 receptor agonist (EC50: 0.45 nM) that is used to manage intraocular pressure associated with open-angle glaucoma or ocular hyperten...
T68114L Nardeterol HCl Nardeterol HCl(73865-18-6 Free base) Adrenergic Receptor
Nardeterol HCl is a β-adrenergic receptor partial agonist used in the study of the central nervous system.CAS 번호13460-73-83-4
T23397 ST 91 Others , Adrenergic Receptor
ST-91 is an agonist of α2-adrenoceptor with a mixed α-adrenergic receptor type/subtype selection profile.
T31750 Faxeladol EM906,GCR 9905,EM 906,GCR-9905,EM-906,GCR9905 5-HT Receptor , Opioid Receptor , Adrenergic Receptor
Faxeladol, a potent adrenergic absorption inhibitor and serotonin reuptake inhibitor, is a small-molecule Opioid receptor agonist that can be used to study neurological disorders.
T8810 Terbutaline Adrenergic Receptor
Terbutaline is a short-acting agonist of β2-adrenergic receptor (β2-AR) . It is an active metabolite of bambuterol
T7164 Levalbuterol tartrate Levosalbutamol tartrate Adrenergic Receptor
Levalbuterol tartrate (Levosalbutamol tartrate) is the β2-adrenergic receptor agonist,and is used to treatment of asthma.
T8358 Fenoterol Adrenergic Receptor
Fenoterol is an agonist of β2-adrenergic receptor It is classed as sympathomimetic beta agonist and asthma medication.
T5954 Methyldopa hydrate Alpha-Methyldopa Sesquihydrate,L-(-)-α-Methyldopa hydrate,MK-351 hydrate,Methyldopa Sesquihydrate Dopamine Receptor , Adrenergic Receptor
Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension. It inhibits the sympathetic nervous system, decreases production of dopamine, ...
T22612 BMY-14802 hydrochloride BMS 181100 hydrochloride,BMY-14802-1,BMY 14802 hydrochloride Sigma receptor , 5-HT Receptor , Adrenergic Receptor
BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 nM) with antipsychotic effects. BMY-14802 hydrochloride is an agonist of the α1-adrenergic receptor and 5-HT1A.
T0290 Tizanidine hydrochloride Tizanidine HCl,DS 103-282 Adrenergic Receptor
Tizanidine hydrochloride (Tizanidine HCl), an α2-adrenergic receptor agonist, inhibits neurotransmitter release from CNS noradrenergic neurons.
T11318 Dopexamine hydrochloride FPL60278AR Adrenergic Receptor
Dopexamine hydrochloride (FPL60278AR) is a β2-adrenergic receptor agonist. Dopexamine can attenuate the inflammatory response and protect against organ injury in the absence of significant effects on hemodynamics or regi...
T22871 Ipsapirone 5-HT Receptor
Ipsapirone is a partial agonist of 5-HT1A receptor and produces an inhibitory effect on 5-HT2 and the α1-adrenergic function at high doses.
T10952 Dabuzalgron Ro 115-1240 Apoptosis , Adrenergic Receptor
Dabuzalgron (Ro 115-1240) is an orally active selective alpha-1A adrenergic receptor agonist used to treat urinary incontinence. Dabuzaron prevents cardiotoxicity caused by doxorubicin by maintaining mitochondrial functi...
T3277 Tulobuterol hydrochloride Lobuterol,Hokunalin,Berachin Influenza Virus , Adrenergic Receptor , Antibiotic
Tulobuterol hydrochloride (Hokunalin) is a long-acting beta2-adrenergic receptor agonist.
T3046 BMY 7378 dihydrochloride BMY7378 HCl Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor
BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.
T21447 Tolazoline Priscol,Priscoline,Pridazole,Divascol,Vasimid,Benzalolin Adrenergic Receptor
Tolazoline (Benzalolin), a non-selective competitive α-adrenergic receptor antagonist, is used as a vasodilator to treat spasms of peripheral blood vessels. It has also been used successfully as an antidote to reverse th...
T6703 Tetrahydrozoline hydrochloride Murine Plus,Tetryzoline hydrochloride,Tyzine,Tetrahydrozoline HCl Adrenergic Receptor
Tetrahydrozoline hydrochloride (Murine Plus) is an imidazoline derivative with alpha receptor agonist activity.
T22029 AL 34662 5-HT Receptor , Adrenergic Receptor
AL 34662 is a selective and potent 5-HT2A receptor agonist with IC50s of 0.77 nM and 1.5 nM for rat and human 5-HT2 receptors, respectively.AL 34662 is also a low affinity α-1D adrenergic agonist, with an EC50 of 0.4 μM....
T2631 WAY-100635 Monomaleate Dopamine Receptor , 5-HT Receptor
WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM. It is also a dopamine D4 receptor agonist with pIC50 values of 8.9 and 6.6 for 5-HT1A ...
T1735 Lurasidone hydrochloride Lurasidone HCl,SM-13496 (Hydrochloride),SM-13496 Dopamine Receptor , 5-HT Receptor , Norepinephrine
Lurasidone hydrochloride (Lurasidone HCl) is a thiazole derivative and atypical antipsychotic agent that functions as a dopamine D2 receptor antagonist; serotonin 5-HT2 receptor antagonist, serotonin 5-HT7 receptor antag...
T12970 Solabegron GW 427353 Adrenergic Receptor
Solabegron (GW 427353) is a selective agonist of β3-adrenergic receptor, stimulating cAMP accumulation in Chinese hamster ovary cells expressing the human β3-AR(EC50 : 22 nM). It is used for treatment of overactive bladd...
T6466 Dexmedetomidine hydrochloride Precedex,(+)-Medetomidine hydrochloride,(S)-Medetomidine hydrochloride,Dexmedetomidine HCl Adrenergic Receptor
Dexmedetomidine hydrochloride (Precedex) is an imidazole derivative that is an agonist of the adrenergic alpha-2 receptor. It is closely-related to MEDETOMIDINE, which is the racemic form of this compound.
T23557 Talibegron hydrochloride ZD2079 hydrochloride,ZD 2079 Adrenergic Receptor
Talibegron hydrochloride (ZD2079 hydrochloride) is an β3 adrenergic receptor agonist with a pD2 of 3.72 on phenylephrine-preconstricted rat mesenteric artery. Relaxes rat mesenteric artery and isolated aorta in vitro. In...
T26666 ASM-024 AChR
ASM-024, a potent nicotinic receptor agonist, is a small molecule synthetic piperazine compound that promotes different targets and signaling pathways of β2-adrenergic receptors mediating smooth muscle relaxation, and is...
T68129L1 Picumeterol FA Picumeterol FA(130641-36-0 Free base) Adrenergic Receptor
picumeterol FA is a potent and selective β2-adrenergic receptor agonist. In in vitro and in vivo tests, picumeterol FA produces long-lasting airway smooth muscle relaxation. picumeterol FA is a pure R-enantiomer and can ...
T38192 Unifiram Others
Unifiram is a nootropic agent.1It increases acetylcholine (ACh) release in the rat cerebral cortexin vivoand induces a long-lasting increase in the amplitude of field excitatory postsynaptic potentials (fEPSPs) in the ra...
T24670 Protokylol JB-251,Protokylolum,JB 251,JB251,Protoquilol
Protokylol is a β-adrenergic receptor agonist.
T25003 Acrinor H 835
Acrinor is a adrenergic beta receptor agonist.
T28885 Sunepitron HCl CP 93,393,CP93,393,CP-93393,CP93393,CP 93393,CP-93,393
Sunepitron is a combined α2-adrenergic receptor antagonist and 5-HT1A receptor agonist.
T11512 Guanoxabenz Hydroxyguanabenz Others
T23281 RWJ 52353 Others
α2D adrenergic receptor agonist
T26651 ARC-239 ARC239,AR C 239,AR C239,AR C-239
ARC-239 is an agonist of α2-adrenergic receptor.

Compounds

Salmeterol
T12829
Synonym: GR33343X
Target: Adrenergic Receptor
Carazolol
T3284
Synonym: Conducton,Suacron
Target: Adrenergic Receptor
Terbutaline Sulfate
T1584
Synonym: Terbutaline hemisulfate
Target: Antibacterial, Adrenergic Receptor, Antibiotic
Isoetharine mesylate salt
T4983
Synonym: Isoetarine mesilate
Target: Others, Adrenergic Receptor
Salmeterol Xinafoate
T6653
Synonym: Salmetedur,GR 33343X xinafoate,Arial
Target: HIV Protease, Adrenergic Receptor
ZK-90055 hydrochloride
T13403
Synonym: ZK 90055 hydrochloride,ZK90055 hydrochloride
Target: Adrenergic Receptor
Mapenterol hydrochloride
T40622
Synonym:
Target: Adrenergic Receptor
Guanabenz Acetate
T6522
Synonym: Wy8678 acetate,BR-750,Wytensin
Target: Adrenergic Receptor
Procaterol hydrochloride
T4548
Synonym:
Target: Adrenergic Receptor
LY377604
T15819
Synonym:
Target: Adrenergic Receptor
Tizanidine
T7065
Synonym:
Target: Adrenergic Receptor
Romifidine
T26119
Synonym: Romifidinum
Target:
AR-08
T10052
Synonym:
Target: Adrenergic Receptor
Tolnapersine TFA
T68023L
Synonym: Tolnapersine TFA(70312-00-4 Free base)
Target: Dopamine Receptor, Adrenergic Receptor
Rafabegron
T34256
Synonym: TAK-677,TAK677,AD9677,AD-9677,TAK 677,AD 9677
Target: Adrenergic Receptor
Salbutamol hemisulfate
T6652
Synonym: Ventolin Sulfate,Albuterol,Salbutamol Sulfate,Bronchospray,Albuterol Sulfate
Target: Adrenergic Receptor, Autophagy
Milveterol HCl
T33386
Synonym: Milveterol,GSK-159797,GSK 159797,GSK159797
Target: Adrenergic Receptor
Apraclonidine hydrochloride
T21371
Synonym: Iopidine,ALO 2145,Apraclonidina,P-aminoclonidine,4-Aminoclonidine,Apraclonidine HCl,Apraclonidinum
Target: Adrenergic Receptor
Brimonidine Tartrate
T6422
Synonym: AGN190342 tartrate,304 tartrate,AGN190342 (tartrate),UK 14304 (tartrate),UK14304 tartrate
Target: Adrenergic Receptor
Nardeterol HCl
T68114L
Synonym: Nardeterol HCl(73865-18-6 Free base)
Target: Adrenergic Receptor
ST 91
T23397
Synonym:
Target: Others, Adrenergic Receptor
Faxeladol
T31750
Synonym: EM906,GCR 9905,EM 906,GCR-9905,EM-906,GCR9905
Target: 5-HT Receptor, Opioid Receptor, Adrenergic Receptor
Terbutaline
T8810
Synonym:
Target: Adrenergic Receptor
Levalbuterol tartrate
T7164
Synonym: Levosalbutamol tartrate
Target: Adrenergic Receptor
Fenoterol
T8358
Synonym:
Target: Adrenergic Receptor
Methyldopa hydrate
T5954
Synonym: Alpha-Methyldopa Sesquihydrate,L-(-)-α-Methyldopa hydrate,MK-351 hydrate,Methyldopa Sesquihydrate
Target: Dopamine Receptor, Adrenergic Receptor
BMY-14802 hydrochloride
T22612
Synonym: BMS 181100 hydrochloride,BMY-14802-1,BMY 14802 hydrochloride
Target: Sigma receptor, 5-HT Receptor, Adrenergic Receptor
Tizanidine hydrochloride
T0290
Synonym: Tizanidine HCl,DS 103-282
Target: Adrenergic Receptor
Dopexamine hydrochloride
T11318
Synonym: FPL60278AR
Target: Adrenergic Receptor
Ipsapirone
T22871
Synonym:
Target: 5-HT Receptor
Dabuzalgron
T10952
Synonym: Ro 115-1240
Target: Apoptosis, Adrenergic Receptor
Tulobuterol hydrochloride
T3277
Synonym: Lobuterol,Hokunalin,Berachin
Target: Influenza Virus, Adrenergic Receptor, Antibiotic
BMY 7378 dihydrochloride
T3046
Synonym: BMY7378 HCl
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor
Tolazoline
T21447
Synonym: Priscol,Priscoline,Pridazole,Divascol,Vasimid,Benzalolin
Target: Adrenergic Receptor
Tetrahydrozoline hydrochloride
T6703
Synonym: Murine Plus,Tetryzoline hydrochloride,Tyzine,Tetrahydrozoline HCl
Target: Adrenergic Receptor
AL 34662
T22029
Synonym:
Target: 5-HT Receptor, Adrenergic Receptor
WAY-100635 Monomaleate
T2631
Synonym:
Target: Dopamine Receptor, 5-HT Receptor
Lurasidone hydrochloride
T1735
Synonym: Lurasidone HCl,SM-13496 (Hydrochloride),SM-13496
Target: Dopamine Receptor, 5-HT Receptor, Norepinephrine
Solabegron
T12970
Synonym: GW 427353
Target: Adrenergic Receptor
Dexmedetomidine hydrochloride
T6466
Synonym: Precedex,(+)-Medetomidine hydrochloride,(S)-Medetomidine hydrochloride,Dexmedetomidine HCl
Target: Adrenergic Receptor
Talibegron hydrochloride
T23557
Synonym: ZD2079 hydrochloride,ZD 2079
Target: Adrenergic Receptor
ASM-024
T26666
Synonym:
Target: AChR
Picumeterol FA
T68129L1
Synonym: Picumeterol FA(130641-36-0 Free base)
Target: Adrenergic Receptor
Unifiram
T38192
Synonym:
Target: Others
Protokylol
T24670
Synonym: JB-251,Protokylolum,JB 251,JB251,Protoquilol
Target:
Acrinor
T25003
Synonym: H 835
Target:
Sunepitron HCl
T28885
Synonym: CP 93,393,CP93,393,CP-93393,CP93393,CP 93393,CP-93,393
Target:
Guanoxabenz
T11512
Synonym: Hydroxyguanabenz
Target: Others
RWJ 52353
T23281
Synonym:
Target: Others
ARC-239
T26651
Synonym: ARC239,AR C 239,AR C239,AR C-239
Target:
1 2 3
カタログ番号 製品名 別名 ターゲット
T6688 Synephrine hydrochloride Oxedrine hydrochloride,Synephrine HCl Endogenous Metabolite , Adrenergic Receptor
Synephrine hydrochloride (Oxedrine hydrochloride) is an agonist that acts on sympathomimetic α-adrenergic receptor (AR).
T0453 Phenylephrine hydrochloride NCI-c55641,Phenylephrine HCl,(R)-(-)-Phenylephrine hydrochloride Endogenous Metabolite , Adrenergic Receptor
Phenylephrine hydrochloride (NCI-c55641) is a selective agonist of the α1-adrenergic receptor.
T4429 Rauwolscine hydrochloride Corynanthidine hydrochloride,α-Yohimbine hydrochloride,Isoyohimbine hydrochloride Adrenergic Receptor
Rauwolscine hydrochloride (Isoyohimbine hydrochloride) , a natural alkaloid, is a specific and reversible α2-adrenergic receptor antagonist (Ki: 12 nM) [1]. It is a stereoisomer of yohimbine, which potently antagonizes b...
T6662 Scopine 6,7-Epoxytropine Adrenergic Receptor
Scopine (6,7-Epoxytropine), the metabolite of anisodine, is an α1-adrenergic receptor agonist used in the therapy of acute circulatory shock.
TN1465 Cannabigerol NOS , 5-HT Receptor , ROS
Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; also binds to the CB2 receptor; it can relieve interocular pressur...
T6519 Gramine NSC 16892,Donaxine Adiponectin receptor , Reverse Transcriptase , Adrenergic Receptor
Gramine (Donaxine), a natural indole alkaloid, present in several plant species, acts as an active adiponectin receptor (AdipoR) agonist, with IC50s of 3.2 and 4.2 μM for AdipoR2 and AdipoR1, respectively. Gramine is als...
T8149 Dobutamine hydrochloride Dobutamine (hydrochloride) Adrenergic Receptor
Dobutamine hydrochloride (Dobutamine (hydrochloride)) is a catecholamine that acts as a β-adrenergic receptor agonist with potent positive inotropic effects.
T60245 Norepinephrine hydrochloride
Norepinephrine hydrochloride (Levarterenol hydrochloride) is a β1 -selective agonist of the adrenergic receptor with EC 50 of 5.37 μM [1].

Recombinant Proteins

カタログ番号 製品名 Species Expression System
TMPJ-00983 ARRB1 Protein, Human, Recombinant (His) Human E. coli
β-Arrestin-1 (ARRB1) is a cytoplasmic protein that belongs to the arrestin family. ARRB1 is expressed at high levels in peripheral blood leukocytes and the central nervous system. ARRB1 regulates agonist-mediated G-prote...
TMPH-02540 GRK2 Protein, Mouse, Recombinant (His & SUMO) Mouse E. coli
Specifically phosphorylates the agonist-occupied form of the beta-adrenergic and closely related receptors, probably inducing a desensitization of them. Key regulator of LPAR1 signaling. Competes with RALA for binding to...